BRD4 Inhibitor-10
BRD4 Inhibitor-10
CAS: 1660117-38-3
Molecular Formula: C25H27N5O2
BRD4 Inhibitor-10 - Names and Identifiers
BRD4 Inhibitor-10 - Physico-chemical Properties
| Molecular Formula | C25H27N5O2 |
| Molar Mass | 429.51 |
BRD4 Inhibitor-10 - Reference Information
| biological activity | BI 894999 is a potent and selective BET inhibitor, the binding of acetylated histones was inhibited by BRD4-BD1 and BRD4-BD2, corresponding to IC50 values of 5 nM and 41 nM, respectively. BI 894999 is highly selective for BRD2/3/4 and BRDT (Kd 0.49-1.6 nM) with at least 200-fold selectivity over BRD4-BD1. |
| Target | Value |
| BET () | |
| BRD4-BD1 (Cell-free assay) | 5 nM |
| BRD4-BD2 (Cell-free assay) | 41 nM |
Last Update：2024-04-10 22:29:15
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Product Name: BRD4 Inhibitor-10 Visit Supplier Webpage Request for quotationCAS: 1660117-38-3
Tel: 18301782025
Email: 3008007409@qq.com
Mobile: 18021002903
QQ: 3008007409
Wechat: 18301782025
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